ID |
Reference |
Source Clone name |
Sequence |
Motif |
Target-tumor |
Target-cell |
Teceptors-biomarker |
Phage/Library |
In vitro/Ex vivo |
In vivo |
Homing/targeting |
Payloads |
Patent |
1017 | Liu S et al. Acta Pharmacol Sin. 2011 Jan;32(1):79-88. | Bombesin | QRLGNQWAVGHLM | NA | Lung, gastric cancer, Neuroblastoma | NA | NA | NA | MCF-7, DU145, A375 HeLa, A875, M14, A549, ZR-75-30, Raji, NB4, K562 cell lines | Eight-week-old female nude mice with MCF-7 xenograft | Homing | MG2 peptide | NA |
1049 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 3 | VPWXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1050 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone5 | GRDS | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1051 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 2 | RGEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1052 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone7 | RGDPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1053 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone8 | WXEPAYQGRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1054 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone9 | WXEPAYNGRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1055 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone10 | RGEPAYQGRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1056 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone11 | RGDPAYQGRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC, Micelle | NA |
1057 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone12 | RGEPAYNGRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1058 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 13 | RGDPAYNGRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1059 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone14 | WXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1060 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone15 | AXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1061 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone16 | WAEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1062 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone17 | WXAPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1063 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone18 | WXEAAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC, Micelle | NA |
1064 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 19 | WXEPAAQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1065 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 20 | WXEPAYARFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1066 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone21 | WXEPAYQAFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1067 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone22 | WXEPAYQAAL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1068 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone23 | WXEPAYQAFA | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1069 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone24 | EXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1070 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone25 | LXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1071 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone26 | KXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1072 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone27 | QXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1073 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 28 | YXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1074 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 29 | FXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1075 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 30 | F*XEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1076 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 31 | FXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1077 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 32 | WEEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1078 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 33 | WLEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1079 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 34 | WIEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1080 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 35 | WKEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1081 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 36 | WQEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1082 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 37 | WTEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1083 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 38 | WXEPAYQREL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1084 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 39 | WXEPAYQRLL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1085 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 40 | WXEPAYQRKL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1086 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 41 | WXEPAYQRQ | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1087 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 42 | WXEPAYQRYL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1088 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 43 | WXEPAYQRF*L | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1089 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 44 | WXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1090 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 45 | WXEPAYQRRE | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1091 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 46 | WXEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1092 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 47 | WXEPAYQRFK | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1093 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 48 | WXEPAYQRFQ | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1094 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 49 | WXEPAYQRFT | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1095 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 50 | WXEPAYQRFF | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1096 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 51 | XEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1097 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 52 | EEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1098 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | Clone 53 | LEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1099 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | LEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1100 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | KEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1101 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | QEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1102 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | TEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1103 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQREL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1104 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRLL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1105 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRKL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1106 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRQL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1107 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRYL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1108 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRF*L | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1109 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1110 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRFE | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1111 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRFL | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1112 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRFK | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1113 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRFQ | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1114 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRFT | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1115 | Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41. | NA | XEPAYQRFF | NA | Breast cancer | NA | NA | NA | Human cancer cell line MDA-MB-435 & MCF-7 | NA | Targeting | FITC | NA |
1206 | Shadidi M et al. FASEB J. 2003 Feb;17(2):256-8. | Ph12-1 | WNLPWYYSVSPT | LTVXPW | Breast cancer | NA | NA | M13 phage/ 12 mer peptide library&M13 phage/7 mer peptide library | The breast cancer cell lines SK-BR-3, T47D, MCF-7, PM-, colon cancer cell line HT2933,prostate cancer cell line DU145; lung cancer cell line DMS-273,U87MG cell line, | NA | Targeting | GFP & 6-iodoacetamido | NA |
1401 | Borgne-Sanchez A et al. Cell Death Differ. 2007 Mar;14(3):422-35. | TEAM-VP | GGCRGDMFGC | RGD | Metastiasis in tumor | Angiogenic endothelial cells | Alpha-5 beta- 3 integrins | NA | HUVEC, HMVECd, A375M, MCF-7, MDA-MB-231, HeLa, HT-29, Jurkat, CEM and fresh peripheral blood mononuclear cells (PBMC) | BALB C mice | Homing | FITC, Apoptic peptide | WO96/15811,US 6,458,026 B1 |
1413 | Koolpe M et al. J Biol Chem. 2005 Apr 29;280(17):17301-11. | NA | QEFSPYMGLEFKKH | NA | Breast cancer | NA | Ephrin-B1 | M13 phage / 12-mer peptide library | MCF-7 human breast cancer cells | NA | Targeting | Biotin | NA |
1414 | Koolpe M et al. J Biol Chem. 2005 Apr 29;280(17):17301-11. | NA | QEFSPNLWGLEFQKN | NA | Breast cancer | NA | Ephrin-B2 | M13 phage / 12-mer peptide library | MCF-7 human breast cancer cells | NA | Targeting | Biotin | NA |
1415 | Koolpe M et al. J Biol Chem. 2005 Apr 29;280(17):17301-11. | NA | QEYSPNLWGHEFRSH | NA | Breast cancer | NA | Ephrin-B3 | M13 phage / 12-mer peptide library | MCF-7 human breast cancer cells | NA | Targeting | Biotin | NA |
1473 | Askoxylakis V et al. Clin Cancer Res. 2005 Sep 15;11(18):6705-12. | p160 | VPWMEPAYQRFL | NA | Human breast cancer | Tumor cell | NA | NA | Breast cancer cell line MDA-MB-435,neuroblastoma cell line WAC 2, MCF-7 | Female BALB/c nu/nu mice carrying human breast cancer MDA-MB-435 tumors | Homing | (131)I-labeled and the FITC-labeled | NA |
1753 | Lu ZX et al. Int J Nanomedicine 2011;6:1661-73. | APRPG peptide | APRPG | NA | Breast cancer | Tumor vessel | VEGF | NA | Human breast cancer cell line MCF-7 | BALB/C nude mice (5 weeks of age) | Homing | NA | US 6,753,310 B1 |