ID Reference Source Clone name Sequence Motif Target-tumor Target-cell Teceptors-biomarker Phage/Library In vitro/Ex vivo In vivo Homing/targeting Payloads Patent
1001He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R22CSNIDARACNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cells, H460 CellBALB/ C mice with lung tumorHomingLiposomal doxorubicinUS2010/0233161A1
1002He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.3R5CDPSRGKNCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1003He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R24CPSDLKDACNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1004He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R4CRTTRGTKCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1005He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R8CRMTRNKPCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1006He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R17CRVSRQNKCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1007He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R9CAKIDPELCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1008He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.3R14CGGERGKSCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1049Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 3VPWXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1050Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone5GRDSNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1051Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 2RGEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1052Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone7RGDPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1053Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone8WXEPAYQGRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1054Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone9WXEPAYNGRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1055Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone10RGEPAYQGRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1056Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone11RGDPAYQGRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITC, MicelleNA
1057Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone12RGEPAYNGRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1058Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 13RGDPAYNGRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1059Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone14WXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1060Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone15AXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1061Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone16WAEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1062Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone17WXAPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1063Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone18WXEAAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITC, MicelleNA
1064Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 19WXEPAAQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1065Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 20WXEPAYARFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1066Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone21WXEPAYQAFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1067Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone22WXEPAYQAALNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1068Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone23WXEPAYQAFANABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1069Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone24EXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1070Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone25LXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1071Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone26KXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1072Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone27QXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1073Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 28YXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1074Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 29FXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1075Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 30F*XEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1076Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 31FXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1077Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 32WEEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1078Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 33WLEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1079Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 34WIEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1080Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 35WKEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1081Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 36WQEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1082Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 37WTEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1083Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 38WXEPAYQRELNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1084Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 39WXEPAYQRLLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1085Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 40WXEPAYQRKLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1086Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 41WXEPAYQRQNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1087Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 42WXEPAYQRYLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1088Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 43WXEPAYQRF*LNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1089Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 44WXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1090Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 45WXEPAYQRRENABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1091Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 46WXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1092Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 47WXEPAYQRFKNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1093Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 48WXEPAYQRFQNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1094Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 49WXEPAYQRFTNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1095Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 50WXEPAYQRFFNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1096Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 51XEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1097Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 52EEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1098Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.Clone 53LEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1099Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NALEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1100Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAKEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1101Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAQEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1102Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NATEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1103Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRELNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1104Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRLLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1105Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRKLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1106Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRQLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1107Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRYLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1108Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRF*LNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1109Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1110Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRFENABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1111Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRFLNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1112Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRFKNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1113Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRFQNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1114Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRFTNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1115Ahmed S et al. Anal Chem. 2010 Sep 15;82(18):7533-41.NAXEPAYQRFFNABreast cancerNANANAHuman cancer cell line MDA-MB-435 & MCF-7NATargetingFITCNA
1127Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NANRLKCRAQATHSAAPCIRGYNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1128Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NARQNSCTYSDARRWALCWSGENABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1129Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAQLNSCIHSGDRAIRGCMDWVNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1130Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAKYGLCRDETVFPSHSCTFTGNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1131Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGSPQCPGGFNCPRCDCGAGYNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1132Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGTGSCGYGKLHTGYWCSYFPNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1133Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NANSSSCDTSVVRSTWACILQPNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1134Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAVRAVCTTLKSRGHEECWSLQNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1135Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAVYAQCGVNVRTGRGGCSRLMNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1136Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAVHMNCSWMRVSEGHPCESADNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1137Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGRQGCYEHLWRLIAWCAIFLNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1138Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NALRMTCAFGVAQRSADCALSSNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1139Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NASIVNCSAALTDLPTRCGGNINABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1140Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NACGTRCVRCQNGPEASCEQPLNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1141Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NATPLFCGNHGRQPSPLCMKWDNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1142Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAFTTVCRQPRGHEAIVCGSGKNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1143Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAAPSFCGTAMLGASRYCYSGPNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1144Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGARECESGGPGMRKLCTQINNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1145Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NANNRACFRTSKGNPAECPYLGNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1146Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGSLACQNIVVCVKKQCNALCNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1147Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAKRASCQNPLFSNFFVCGLSENABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1148Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NALPNFCMDTSGRAGPLCMGSENABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1149Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NARHTVCRVSLSSVQGSCSHEYNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1160Zhang L et al. Cancer Res. 2006 Jun 1;66(11):5696-706.LSDCLSDGKRKCNAHuman melanomaLymphatic vesselPodoplanin, Prox-1,LYVE-1 and VEGFR-10T7 phage/CX7C peptide libraryC8161 human melanoma, MDA-MB-435 human breast cancerMice bearing C8161 cells human cancer xenograftsHomingRadioactive indium, proapoptotic peptideUS 2007/0219134A1
1161Zhang L et al. Cancer Res. 2006 Jun 1;66(11):5696-706.NACLDGGRPKCNAHuman melanomaLymphatic vesselPodoplanin,Prox-1,LYVE-1 and VEGFR-10T7 phage/CX7C peptide libraryC8161 human melanoma, MDA-MB-435 human breast cancerMice bearing C8161 cells human cancer xenograftsHomingFluoresceineNA
1162Zhang L et al. Cancer Res. 2006 Jun 1;66(11):5696-706.REA CREAGRKACNAProstrate cancerLymphatic vesselPodoplaninT7 phage/CX7C peptide libraryMDA-MB-435 human breast cancer cell lineTRAMP mice, Nude mice bearing xenogragt from the human prostate cancer cell lines PPC1, M12, DU145, and LNCaPHomingRadioactive indium, proapoptotic peptideUS 2007/0219134A1
1163Zhang L et al. Cancer Res. 2006 Jun 1;66(11):5696-706.AGRCAGRRSAYCNAProstrate cancerLymphatic vesselPodoplaninT7 phage/CX7C peptide libraryMDA-MB-435 human breast cancer cell lineTRAMP miceHomingFluoresceineUS 2007/0219134A1
1164Zhang L et al. Cancer Res. 2006 Jun 1;66(11):5696-706.Lyp-2CNRRTKAGCNACervical CancerLymphatic vesselPodoplaninT7 phage/CX7C peptide libraryMDA-MB-435 human breast cancer cell lineK14-HPV-16 miceHomingFluoresceineUS 2007/0219134A1
1171Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7.P-5m GHGKHKNKGHGKHKNKHGKLung metastassisNAVitronectinNAMDA-MB-231 cellsMice bearing malignant melanoma cell line B16-F10 derived tumorHomingNANA
1172Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7.P-5 (His479—Lys493)HKHGHGHGKHKNKGKHGKBreast cancerNAVitronectinNAMDA-MB-231 cellsNATargetingNANA
1173Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7.P-5n (Lys480—Lys487)KHGHGHGKHGKBreast cancerNAVitronectinNAMDA-MB-231 cellsNATargetingNANA
1174Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7.P-5nKGHHGKHGHGKBreast cancerNAVitronectinNAMDA-MB-231 cellsNATargetingNANA
1175Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7.P-5c (His488—Asn495)HKNKGKKNHGKBreast cancerNAVitronectinNAMDA-MB-231 cellsNATargetingNANA
1238Houimel M et al. Int J Cancer. 2001 Jun 1;92(5):748-55.NAMARSGLNAHuman breast and ovarian adenocarcinomasTumor cellErbB-2NASK-BR-3, MDA-MB-468, OVCAR3NATargeting & further studiedNANA
1239Houimel M et al. Int J Cancer. 2001 Jun 1;92(5):748-55.NAMARAKENAHuman breast and ovarian adenocarcinomasTumor cellErbB-2NASK-BR-3, MDA-MB-468, OVCAR4NATargeting & further studiedNANA
1240Houimel M et al. Int J Cancer. 2001 Jun 1;92(5):748-55.NAMSRTMSNAHuman breast and ovarian adenocarcinomasTumor cellErbB-2NASK-BR-3, MDA-MB-468, OVCAR5NATargeting & further studiedNANA
1272Zhang J et al. Cancer Lett. 2001 Oct 10;171(2):153-64.p160VPWMEPAYQRFLNANeuroblastoma and breast cancerNANAM13 phage /12 mer peptide libraryHuman neuroblastoma cell lines WAC-2, Human breast cancer cell line MDA-MB-435NATargetingFITCNA
1273Zhang J et al. Cancer Lett. 2001 Oct 10;171(2):153-64.p36MLPKPSSFPVPGNANeuroblastoma and breast cancerNANAM13 phage /12 mer peptide libraryHuman neuroblastoma cell lines WAC-2, Human breast cancer cell line MDA-MB-435NATargetingFITCNA
1274Zhang J et al. Cancer Lett. 2001 Oct 10;171(2):153-64.p155HSFLHPWDLFDYNANeuroblastoma and breast cancerNANAM13 phage /12 mer peptide libraryHuman neuroblastoma cell lines WAC-2, Human breast cancer cell line MDA-MB-435NATargetingFITCNA
1275Pasqualini R et al. Cancer Res. 2000 Feb 1;60(3):722-7.NACNGRCVSGCAGRCNABreast cancerNANAM13 phage /CX3CX3CX3C peptide libraryMDA-MB-435 breast cancer cells transfected with APN cDNA.Mice bearing MDA-MB-435 tumorsHomingDoxorubicinWO06067633A2
1276Pasqualini R et al. Cancer Res. 2000 Feb 1;60(3):722-7.NACVLNGRMECNABreast cancerNANAM13 phage /CX3CX3CX3C peptide libraryMDA-MB-435 breast cancer cells transfected with APN cDNA.Mice bearing MDA-MB-435 tumorsHomingDoxorubicinUS 2009/0257951 A1
1312Peletskaya EN et al. J Mol Biol. 1997 Jul 18;270(3):374-84.P30HGRFILPWWYAFSPSW-Y-A-W/F-S-PBreast cancerNAGal beta1 --> 3GalNAc alpha disaccharidef3 Bacteriophage/ 15-mer peptide libraryMDA-MB-435 breast carcinoma cellsNATargetingFITCUS 2004/0010116 A1
1313Peletskaya EN et al. J Mol Biol. 1997 Jul 18;270(3):374-84.P89RFRGLISLSQVYLSPNABreast cancerNAGal beta1 --> 3GalNAc alpha disaccharidef3 Bacteriophage/ 15-mer peptide libraryHuman breast carcinoma cell line MDA-MB-435NATargetingFITCNA
1314Peletskaya EN et al. J Mol Biol. 1997 Jul 18;270(3):374-84.P6ARVSFWRYSSFAPTYNABreast cancerNAGal beta1 --> 3GalNAc alpha disaccharidef3 Bacteriophage/ 15-mer peptide libraryHuman breast carcinoma cell line MDA-MB-435NATargetingNANA
1315Peletskaya EN et al. J Mol Biol. 1997 Jul 18;270(3):374-84.P10GSWYAWSPLVPSAQINABreast cancerNAGal beta1 --> 3GalNAc alpha disaccharidef88 Bacteriophage/15 mer peptide libraryHuman breast carcinoma cell line MDA-MB-435NATargetingFITCNA
1320Drecoll E et al. PLoS One. 2009 May 27;4(5):e5715.F3KDEPQRRSARLSAKPAPPKPEPKPKKAPAKKNAPeritoneal carcinomatosisNucleus of tumor cellsNucleoinNAEMT6, MIAPACA, CMT93, OVCAR3, MDA-MB-435 cell lineMice bearing intra-peritoneal MDA-MB-435 xenograft tumorsHomingBi-DTPA-[F3]2EP1783140A3,US 7,544,767B2
1387Kumar SR et al. Clin Cancer Res. 2007 Oct 15;13(20):6070-9.NAKCCYSLNAHuman breast carcinomaTumor cellErbB-2NAMDA-MB,Human breast carcinoma cell line, Prostate carcinoma cell line (PC-3),K-562 human erythroid leukemia cell lineSCID mice, MDA-MB-435 breast carcinoma cellHoming111In-DOTA, BiotinUS 2010/0061930
1401Borgne-Sanchez A et al. Cell Death Differ. 2007 Mar;14(3):422-35.TEAM-VPGGCRGDMFGCRGDMetastiasis in tumorAngiogenic endothelial cellsAlpha-5 beta- 3 integrinsNAHUVEC, HMVECd, A375M, MCF-7, MDA-MB-231, HeLa, HT-29, Jurkat, CEM and fresh peripheral blood mononuclear cells (PBMC)BALB C miceHomingFITC, Apoptic peptideWO96/15811,US 6,458,026 B1
1454Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.G3-A9PQNSKIPGPTFLDPHP-(C)-G-P-XXX-D(C)-PTumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549 trans, Human breast carcinoma cell line MDA-MB-435, Human prostate carcinoma cell line PC-3M, MDA-MB-435 human breast carcinoma cells on HBME-1 monolayersNATargeting & further studiedNANA
1462Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.G3-C9AYTKCSRQWRTCMTTHNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3M,MDA-MB-435 human breast carcinoma cells on HBME-1 monolayersNATargeting & further studiedNANA
1463Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.G3-C12ANTPCGPYTHDCPVKRP-(C)-G-P-XXX-D(C)-PTumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3M,MDA-MB-435 human breast carcinoma cells on HBME-1 monolayersNATargeting & further studiedNANA
1464Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-C44NISRCTHPFMACGKQSNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide librarySaos2 (derived from a human osteosarcoma),Human breast cancer cell lines BT549, express detectable levels of galectin-3 ,BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3MNATargetingNANA
1465Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-C60PRNICSRRDPTCWTTYNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide librarySaos2 (derived from a human osteosarcoma),Human breast cancer cell lines BT549, express detectable levels of galectin-3 ,BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3MNATargetingNANA
1468Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36.NACVSNPRWKCNAPancreatic islet tumorsTumor vesselEphA4, a receptor for epinephrine-APhage/ CX7C peptide library EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cellsMale C57BL/6/RIP-Tag2 transgenic mice HomingNANA
1469Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36.NACHVLWSTRCNAPancreatic islet tumorsTumor vesselEphA4, a receptor for epinephrine-APhage/ CX7C peptide library EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cellsMale C57BL/6/RIP-Tag2 transgenic mice TargetingNANA
1470Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36.NASWLAYPGAVSYRNAPancreatic islet tumorsTumor vesselEpinephrine-APhage/ CX7C peptide library EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cellsMale C57BL/6/RIP-Tag2 transgenic mice TargetingNANA
1471Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36.NAYSAYPDSVPMMSNAPancreatic islet tumorsTumor vesselEpinephrine-APhage/ CX7C peptide library EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cellsMale C57BL/6/RIP-Tag2 transgenic mice TargetingNANA
1473Askoxylakis V et al. Clin Cancer Res. 2005 Sep 15;11(18):6705-12.p160VPWMEPAYQRFLNAHuman breast cancerTumor cellNANABreast cancer cell line MDA-MB-435,neuroblastoma cell line WAC 2, MCF-7Female BALB/c nu/nu mice carrying human breast cancer MDA-MB-435 tumorsHoming(131)I-labeled and the FITC-labeledNA
1482Yang W et al. Clin Cancer Res. 2008 Sep 1;14(17):5494-502.TMTP1NVVRQGCGXXXXXGCTumor metastasisNANAfUSE5 phage /CX7C peptide libraryPC-3M-1E8, MDA-MB-435S,PG-BE1,MKN-45sciNATargetingNANA
1483Pasqualini R et al. Nat Biotechnol. 1997 Jun;15(6):542-6.NACDCRGDCFCNAMalignant melanomas and breast carcinomaNAAlpha -5 beta-1 integrinPhage /RGD-4CLibraryMDA-MB-435 breast cancer cells, murine B16B15b melanoma,C8161 human melanomaFemale 2-month old BALB/ C miceHomingNANA
1498NANACGNKRTRGCNABreast cancerLymphatic vesselNAT7 phage / random peptide libraryMDA-MB-435 breast carcinoma cell lineHIFko tumor-bearing miceHoming (Phage display clone)NAU.S. Pat. No. 7192921
1683NAClone 11PQRRSARLSANATumor angiogenesisNANucleolinNAHL-60 , MDA-MB-435Nude mice bearing HL-60 tumorsHomingFITCUS 2009/0098633A1
1710NAClone 13CALIIQKNECNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1711NAClone 14CGLILQKNECNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1712NAClone 15CGLIIQRNECNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1713NAClone 16CGLIINKNECNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1714NAClone 17CNAAESSKNCNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1715NAClone 18CNAGESSRNCNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1716NAClone 19CNAGESTKNCNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1717NANACNAGDSSKNCNAMultiple tumorNANANAB16F1 mouse melanoma, Lewis lung carcinoma, C8161 human melanoma, MDA-MB-435 human breast cancer, and PPC-1 human prostate cancer cell lineNATargetingNAUS 2009/0214429 A1
1746Kumar A et al.Biomaterials 2012 Feb;33(4):1180-9.NACRGDKNABreast cancerNANRP-1NAMDA-MB-321 overexpresses Nrp-1 receptor.NATargetingGoldnanoparticlees with therapeutic peptide p12(TSFAEYWNLLSP)US2010/0172835
1747Numata K et al. Macromol Biosci 2012 Jan;12(1):75-82. F3 peptidesKDEPQRRSARLSAKPAPPKPEPKPKKAPAKKNABreast cancerEndothelial cellNucleolinNAMDA-MB-435 melanoma cell line, MDA-MB-231 human breast tumor cell lineNAHomingSilk-based ionic pDNA complexesUS 7,544,767 B2
1748Numata K et al. Macromol Biosci 2012 Jan;12(1):75-82. Lyp1 peptideCGQKRTRGCNABreast cancerNANANAMDA-MB-435 melanoma cell line, MDA-MB-231 human breast tumor cell lineNAHomingSilk-based ionic pDNA complexesUS 2010/0172 835 A1
1756Numata K et al .Bioconjug Chem 2011 Aug 17;22(8):1605-10.F3KDEPQRRSARLSAKPAPPKPEPKPKKAPAKKNABreast tumorTumor vesselNucleolinNAMDA-MB-435 melanoma cell line, MDA-MB-231Mice bearing MDA-MB-231HomingpDNA complexes of silk proteins containing poly(L-lysine)US 7,544,767 B2
1757Numata K et al .Bioconjug Chem 2011 Aug 17;22(8):1605-10.NACGKRKNABreast tumorTumor vesselHeparansulphateNAMDA-MB-435 melanoma cell line, MDA-MB-231Mice bearing MDA-MB-231HomingpDNA complexes of silk proteins containing poly(L-lysine)US 7,723,474 B2
1758Bhojani MS et al .PloS One. 2011;6(7):e22418. Modified F3KDEPQRRSARLSAKPAPPKPEPKPKKAPAKKCNABreast tumorTumor vesselNucleolinNAMDA-MB-435 melanoma cell lineNude Mice bearing MDA-MB-435HomingRadio idionated maleimide conjugating groupUS 2005/0196343 A1