| ID |
Reference |
Source Clone name |
Sequence |
Motif |
Target-tumor |
Target-cell |
Receptors-biomarker |
Phage/Library |
In vitro/Ex-vivo |
In vivo |
Homing/targeting |
Payloads |
Patent |
| 1171 | Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7. | P-5m GHGKHKNK | GHGKHKNK | HGK | Lung metastassis | NA | Vitronectin | NA | MDA-MB-231 cells | Mice bearing malignant melanoma cell line B16-F10 derived tumor | Homing | NA | NA |
| 1172 | Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7. | P-5 (His479â€â€Lys493) | HKHGHGHGKHKNKGK | HGK | Breast cancer | NA | Vitronectin | NA | MDA-MB-231 cells | NA | Targeting | NA | NA |
| 1173 | Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7. | P-5n (Lys480â€â€Lys487) | KHGHGHGK | HGK | Breast cancer | NA | Vitronectin | NA | MDA-MB-231 cells | NA | Targeting | NA | NA |
| 1174 | Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7. | P-5n | KGHHGKHG | HGK | Breast cancer | NA | Vitronectin | NA | MDA-MB-231 cells | NA | Targeting | NA | NA |
| 1175 | Kawasaki M et al. J Biol Chem. 2003 Dec 5;278(49):49301-7. | P-5c (His488â€â€Asn495) | HKNKGKKN | HGK | Breast cancer | NA | Vitronectin | NA | MDA-MB-231 cells | NA | Targeting | NA | NA |
| 1176 | Joyce JA et al. Cancer Cell. 2003 Nov;4(5):393-403. | RGR | CRGRRST | RGRRS, RGRR | Pancreatic islet carcinoma | Endothelial cellor pericytes | NA | T7 phage/CX7C peptide library | NA | Prototypical mouse model of multistage tumorigenesis, RIP1-Tag2 transgenic model of islet cell carcinoma and K14-HPV16 mice | Homing | NA | WO05041882A2,US20050245445A1 |
| 1177 | Joyce JA et al. Cancer Cell. 2003 Nov;4(5):393-403. | RSR | CRSRKG | CRSR-GCRSR-G | Pancreatic islet carcinoma | Endothelial cellor pericytes | NA | T7 phage/CX7C peptide library | NA | Prototypical mouse model of multistage tumorigenesis, RIP1-Tag2 transgenic model of islet cell carcinoma and K14-HPV16 mice | Homing | NA | US 2005/0245445A1 |
| 1178 | Joyce JA et al. Cancer Cell. 2003 Nov;4(5):393-403. | KAA | CKAAKNK | CKA-K | Pancreatic islet carcinoma | Endothelial cellor pericytes | NA | T7 phage/CX7C peptide library | NA | Prototypical mouse model of multistage tumorigenesis, RIP1-Tag2 transgenic model of islet cell carcinoma and K14-HPV16 mice | Homing | NA | US 2005/0245445A1 |
| 1179 | Joyce JA et al. Cancer Cell. 2003 Nov;4(5):393-403. | KAR | CKGAKAR | CKGAKA, AKAR, GAKAR | Pancreatic islet carcinoma | Endothelial cellor pericytes | NA | T7 phage/CX7C peptide library | NA | Prototypical mouse model of multistage tumorigenesis, RIP1-Tag2 transgenic model of islet cell carcinoma and K14-HPV16 mice | Homing | NA | US 2010/0076175A1 |
| 1180 | Joyce JA et al. Cancer Cell. 2003 Nov;4(5):393-403. | VGVA | FRVGVADV | F-VGVADV, RVGV | Pancreatic islet carcinoma | Endothelial cellor pericytes | NA | T7 phage/CX7C peptide library | NA | Prototypical mouse model of multistage tumorigenesis, RIP1-Tag2 transgenic model of islet cell carcinoma and K14-HPV16 mice | Homing | NA | US 2005/0245445A1 |
| 1181 | Joyce JA et al. Cancer Cell. 2003 Nov;4(5):393-403. | EYQ | CEYQLDVE | CEYQL, YQLDV, YQLDV | Pancreatic islet carcinoma | Endothelial cellor pericytes | NA | T7 phage/CX7C peptide library | NA | Prototypical mouse model of multistage tumorigenesis, RIP1-Tag2 transgenic model of islet cell carcinoma and K14-HPV16 mice | Homing | NA | US 2005/0245445 A1 |
| 1182 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CSRPRRSEC | NA | Epidermal squamous cell cancers | Vasculature of earlier stage dysplasias | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | WO0503949542,US20050245445A1 |
| 1183 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CGKRK | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | US 2006/0002854A1 |
| 1184 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CDTRL | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | US 2006/0002854A1 |
| 1185 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CGTKRKC | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | NA |
| 1186 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CDTAVVEGL | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | US 2011/0003848 A1 |
| 1190 | Rafii S et al. Cancer Cell. 2003 Nov;4(5):331-3. | NA | CRSRKG | NA | Pancreatic tumor | Tumor vessel | NA | T7 phage /9-mer cyclic (CX7C) peptide library | NA | RIP-Tag2 pancreatic tumors in murine model | Homing | NA | US 7,598,341 B2 |
| 1191 | Rafii S et al. Cancer Cell. 2003 Nov;4(5):331-3. | NA | CEYQLDVE | NA | Pancreatic tumor | Tumor vessel | NA | T7 phage /9-mer cyclic (CX7C) peptide library | NA | RIP-Tag2 pancreatic tumors in murine model | Homing | NA | US 7,598,341 B2 |
| 1192 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | RPMrel peptide | CPIEDRPMC | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29, Human biopsies | NA | Targeting | Mtochondrial toxin (KLAKLAK)2 | US 7,452,965b2 |
| 1193 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | PIEDRPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1194 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | PIDERPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1195 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | ALRDRPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1196 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | PMMRQRPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1197 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | PLASRPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1198 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | PEKFRPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1199 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | VPEQRPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1200 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | DLPMHPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1201 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | QFQSQPM | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1202 | Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44. | NA | QPPMEYS | NA | Colorectal cancer | Tumor cell | NA | M13 phage/ CX7C peptide library | Colon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29 | NA | Targeting | NA | NA |
| 1203 | Pastorino F et al. Cancer Res. 2003 Nov 1;63(21):7400-9. | NA | NGRSL | NGR | Neuroblastoma | Endothelial cell | Aminopeptidase N | NA | Five human NB cell lines GI-ME-N, GI-LI-N, HTLA-230, IMR-32, and SH-SY5Y, KS1767 cells | Orthotopic neuroblastoma (NB) xenografts in SCID mice | Homing | Liposomal doxorubicin (NGR-SL[DXR]) | US 2009/0092663A1 |
| 1204 | Pan W et al. J Biol Chem. 2003 Jul 25;278(30):27820-7. | NA | MTQMIS | PL(G/P/A)↓L(R/M) | Multiple tumor | NA | MMP-11 proteinase | M13 phage/ 6 mer peptide library | ELISA assay with MMP-11 as substrate | NA | Targeting | NA | NA |
| 1205 | Pan W et al. J Biol Chem. 2003 Jul 25;278(30):27820-7. | NA | TALSPQ | NA | Multiple tumor | NA | MMP-11 proteinase | M13 phage/ 6 mer peptide library | ELISA assay with MMP-11 as substrate | NA | Targeting | NA | NA |
| 1261 | NA | NA | CGSLVRC | GSL | Breast tumor | Tumor cell | NA | Phagedisplaying an Arg  Gly  Asp ( RGD )  containing peptide | NA | Mice bearing human 435 breast carcinoma | Homing | Doxorubicin | US 2003/0152578 A1 |
| 1494 | NA | NA | CTTHWGFTLC | HWGF | Multiple tumor | NA | MMP2 | CX 9 library | The HT1080 fibrosarcoma cells , C8161 melanoma cells and Eahy926 cells (derivative of HUVEC) | Mice bearing human breast carcinomas(MDA-B-435) | Homing | NA | US 6,624,144 B1 |
| 1495 | NA | NA | CRRHWGFEFC | HWGF | Multiple tumor | NA | MMP9 | CX 9 library | The HT1080 fibrosarcoma cells , C8161 melanoma cells | NA | Targeting | NA | US 6,624,144 B1 |
| 1692 | NA | Clone 11 | AGTRMSWEV | NA | Tumor angiogenesis | NA | NA | M13 phage /10 mer peptide library | NA | Mice | Homing | NA | US6528481 |